SCHEMBL5014295

SCHEMBL5014295

CC1CN(c2c(CO)cc(C(=O)S)c(F)c2F)CC(C)O1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
KDM4E B2RXH2 4/20 0.36
HTT P42858 1/20 0.36
ALDH1A1 P00352 8/20 0.35
NPSR1 Q6W5P4 2/20 0.35
HPGD P15428 4/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GAA P10253 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2C19 P33261 2/20 0.32
POLB P06746 1/20 0.32
USP30 Q70CQ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3069796 0.89 KDM4E (0.38) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL2309750 0.89 TSHR (0.38) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL2307645 0.85 TSHR (0.36) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL5014297 0.84 KDM4E (0.36) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL2305888 0.82 ALDH1A1 (0.45) KDM4EALDH1A1NPSR1HPGDTDP1
Hydrochloric Acid SCHEMBL5012175 0.79 MAPT (0.34) TSHRKDM4EHTT
SCHEMBL3653239 0.79 KDM4E (0.33) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL3066491 0.79 KDM4E (0.36) TSHRKDM4EHTTALDH1A1NPSR1
SCHEMBL2308459 0.78 KDM4E (0.39) TSHRKDM4EHTTALDH1A1TDP1
SCHEMBL2310229 0.78 SCN9A (0.40) KDM4EHTTALDH1A1NPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888597-A2 ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2008-02-20 EP disclosed
WO-2006120563-A2 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2006-11-16 WO disclosed