SCHEMBL5015040

SCHEMBL5015040

Oc1cccc2sc(N3CCN(Cc4ccc(C(F)(F)F)cc4)CC3)nc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
NPC1 O15118 3/20 0.50
CASP1 P29466 1/20 0.47
CASP4 P49662 1/20 0.47
CASP5 P51878 1/20 0.47
PPARG P37231 1/20 0.46
PPARD Q03181 1/20 0.46
PPARA Q07869 1/20 0.46
PANK3 Q9H999 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ACHE P22303 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5015038 0.89 RAB9A (0.50) RAB9AMEN1KMT2ANPC1CASP1
SCHEMBL5063385 0.86 RAB9A (0.67) RAB9AMEN1KMT2ANPC1ALDH1A1
SCHEMBL2094261 0.83 RPS6KB1 (0.44) RAB9AMEN1KMT2ANPC1PANK3
SCHEMBL5013361 0.81 MEN1 (0.52) RAB9AMEN1KMT2ANPC1PANK3
SCHEMBL2096584 0.77 SCD (0.46) RAB9ANPC1SMN1; SMN2L3MBTL1MAPT
SCHEMBL5063380 0.75 RAB9A (0.67) RAB9AMEN1KMT2ANPC1ALDH1A1
SCHEMBL2091153 0.73 SMN1; SMN2 (0.68) RAB9ANPC1PPARGKDM4EALDH1A1
SCHEMBL2094258 0.72 RPS6KB1 (0.44) RAB9ANPC1PANK3SMN1; SMN2L3MBTL1
SCHEMBL10219646 0.72 PPARD (0.62) RAB9AMEN1KMT2ANPC1PPARG
SCHEMBL10219602 0.72 PPARD (0.65) RAB9AMEN1KMT2ANPC1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed