SCHEMBL5015646

SCHEMBL5015646

COc1ccc2c(C(=O)O)cc3c(c2c1)=C[N]C(=O)C=3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 12/20 0.47
ALDH1A1 P00352 9/20 0.47
POLB P06746 5/20 0.47
HPGD P15428 5/20 0.47
HSD17B10 Q99714 2/20 0.47
GAA P10253 3/20 0.46
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA3 P07451 2/20 0.46
CA5A P35218 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
CA5B Q9Y2D0 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CA4 P22748 1/20 0.46
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5024158 0.79 TP53 (0.41) KDM4EHSD17B10LMNASMN1; SMN2
SCHEMBL5025775 0.72 HSD17B1 (0.45) KDM4EALDH1A1POLBHSD17B10SMN1; SMN2
SCHEMBL28018438 0.69 KDM4E (0.59) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL24895093 0.66 LMNA (0.55) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL10390929 0.66 LMNA (0.59) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL26965977 0.66 KDM4E (0.81) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL16832123 0.66 KDM4E (0.58) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL21070811 0.65 LMNA (0.54) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL5009698 0.65 KDM4E (0.54) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL15129579 0.64 KDM4E (0.73) KDM4EALDH1A1POLBHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904449-A2 INHIBITORS OF CHECKPOINT KINASES Merck & Co., Inc. (US) 2008-04-02 EP disclosed
WO-2007008502-A2 INHIBITORS OF CHECKPOINT KINASES MERCK & CO., INC. (US) 2007-01-18 WO disclosed