SCHEMBL5017643

SCHEMBL5017643

NC(=O)C1(c2ccc(C(=S)Nc3ccc(Oc4ccnc5ccsc45)c(F)c3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.56
KDR P35968 13/20 0.56
AXL P30530 1/20 0.40
RET P07949 1/20 0.40
KIT P10721 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562834 0.80 MET (0.70) METKDR
SCHEMBL12376838 0.76 MET (0.67) METKDRAXLRETKIT
SCHEMBL5017641 0.73 MET (0.60) METKDR
SCHEMBL2284919 0.73 MET (0.87) METKDR
SCHEMBL2289171 0.72 MET (0.72) METKDRAXLPDGFRA
SCHEMBL307620 0.72 MET (1.00) METKDR
SCHEMBL2277830 0.72 MET (0.64) METKDR
SCHEMBL18516581 0.71 MET (0.64) METKDR
SCHEMBL2277849 0.71 MET (0.67) METKDR
SCHEMBL2282742 0.71 MET (1.00) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904504-A2 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING Methylgene, Inc. (CA) 2008-04-02 EP disclosed
WO-2007054831-A2 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE, INC. (CA) 2007-05-18 WO disclosed