SCHEMBL5019760

SCHEMBL5019760

Cc1cccc(F)c1C(=O)Nc1ccc(C2=C(C3CC3)CCN(c3nnn(C)n3)C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IL2 P60568 6/20 0.38
TNF P01375 1/20 0.37
STIM1 Q13586 1/20 0.37
ORAI1 Q96D31 1/20 0.37
CRACR2A Q9BSW2 5/20 0.36
CHRNA7 P36544 1/20 0.34
KCNH2 Q12809 1/20 0.34
JAK1 P23458 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
C5AR1 P21730 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
BMX P51813 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1781053 0.95 CRACR2A (0.40) IL2TNFSTIM1ORAI1CRACR2A
SCHEMBL5019598 0.89 IL2 (0.40) IL2TNFSTIM1ORAI1CHRNA7
SCHEMBL5019639 0.88 IL2 (0.40) IL2TNFSTIM1ORAI1CHRNA7
SCHEMBL987243 0.85 IL2 (0.43) IL2TNFSTIM1ORAI1CHRNA7
SCHEMBL5019607 0.84 STIM1 (0.42) IL2STIM1ORAI1CRACR2ANPC1
SCHEMBL1782420 0.82 IL2 (0.41) IL2TNFSTIM1ORAI1CHRNA7
SCHEMBL1781986 0.80 IL2 (0.46) IL2JAK1NPC1RAB9A
SCHEMBL5019740 0.80 GAA (0.42) IL2TNFSTIM1ORAI1C5AR1
SCHEMBL5019619 0.79 TYK2 (0.45) IL2JAK1ITGB1ITGA4
SCHEMBL5019662 0.79 IL2 (0.40) IL2STIM1ORAI1CRACR2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064808-A1 TETRAZOLYL - TETRAHYDROPYRIDINE COMPOUNDS FOR INFLAMMATION AND IMMUNE - RELATED USES SYNTA PHARMACEUTICALS CORP (US) 2012-05-18 WO disclosed