SCHEMBL5021040

SCHEMBL5021040

COc1ccc2cc(Br)c(C(C)(F)F)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.44
CYP1A2 P05177 1/20 0.44
HSD17B1 P14061 1/20 0.43
HSD17B2 P37059 1/20 0.43
PTPN1 P18031 5/20 0.43
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.38
GSTP1 P09211 1/20 0.38
PTPN2 P17706 1/20 0.37
NCF1 P14598 1/20 0.37
NPC1 O15118 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5021031 0.79 PTPN1 (0.63) CYP2A6CYP1A2PTPN1KDM4EPTPN2
SCHEMBL5021024 0.79 PTPN1 (0.71) PTPN1PTPN2
SCHEMBL5020990 0.75 PTPN1 (0.51) CYP2A6CYP1A2PTPN1PTPN2
SCHEMBL1042195 0.74 NOTUM (0.54) CYP2A6CYP1A2RAB9A
SCHEMBL5021033 0.74 RELA (0.51) CYP1A2PTPN1
SCHEMBL5021034 0.73 CYP2A6 (0.46) CYP2A6PTPN1RAB9APTPN2NPC1
SCHEMBL23643815 0.73 CYP1A2 (0.52) CYP2A6CYP1A2HSD17B1HSD17B2RAB9A
SCHEMBL29732501 0.73 CYP1A2 (0.52) CYP2A6CYP1A2HSD17B1HSD17B2RAB9A
SCHEMBL14503733 0.73 CYP1A2 (0.52) CYP2A6CYP1A2HSD17B1HSD17B2RAB9A
SCHEMBL14502703 0.72 CA1 (0.47) CYP2A6CYP1A2RAB9AKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168815-B2 Fused aromatic PTP-1B inhibitors KANEQ PHARMA INC. (CA) 2012-05-01 US disclosed