SCHEMBL5021034

SCHEMBL5021034

CC(=O)c1ccc2cc(Br)c(C(C)(F)F)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.46
PTPN1 P18031 8/20 0.46
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
PTPN2 P17706 2/20 0.40
NOTUM Q6P988 1/20 0.40
PTPRC P08575 1/20 0.38
MEN1 O00255 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
KMT2A Q03164 2/20 0.38
KIF11 P52732 1/20 0.37
CA2 P00918 1/20 0.35
ESRRA P11474 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP3A4 P08684 1/20 0.35
PDK2 Q15119 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2691065 0.83 PTPN1 (0.69) PTPN1PTPN2PTPRC
SCHEMBL2692776 0.77 PTPN1 (0.48) CYP2A6PTPN1PTPN2PTPRCMEN1
SCHEMBL5021031 0.76 PTPN1 (0.63) CYP2A6PTPN1ALDH1A1HPGDPTPN2
SCHEMBL15105728 0.74 CYP2A6 (0.69) CYP2A6MAPTALDH1A1HPGDMEN1
SCHEMBL21215857 0.74 CYP2A6 (0.69) CYP2A6MAPTALDH1A1HPGDMEN1
SCHEMBL834744 0.74 CYP2A6 (0.68) CYP2A6MAPTALDH1A1HPGDMEN1
SCHEMBL17056474 0.74 NOTUM (0.68) MAPTNOTUMMEN1NPC1RAB9A
SCHEMBL5021040 0.73 CYP2A6 (0.44) CYP2A6PTPN1PTPN2NPC1RAB9A
SCHEMBL599006 0.72 CYP2A6 (0.79) CYP2A6MAPTALDH1A1HPGDMEN1
SCHEMBL29451111 0.72 CYP2A6 (0.79) CYP2A6MAPTALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168815-B2 Fused aromatic PTP-1B inhibitors KANEQ PHARMA INC. (CA) 2012-05-01 US disclosed