SCHEMBL5023403

SCHEMBL5023403

CCCCC(=O)C=CC(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.50
POLB P06746 1/20 0.48
POLA1 P09884 1/20 0.48
IAPP P10997 2/20 0.46
CES1 P23141 2/20 0.44
CES2 O00748 1/20 0.44
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
ALDH1A1 P00352 2/20 0.43
TP53 P04637 2/20 0.41
FAAH O00519 2/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
SOAT1 P35610 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.40
CA1 P00915 1/20 0.39
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5023396 1.00 TRPA1 (0.50) TRPA1POLBPOLA1IAPPCES1
SCHEMBL29639618 0.91 POLB (0.59) TRPA1POLBPOLA1CES1CES2
SCHEMBL11099789 0.88 TRPA1 (0.60) TRPA1POLBPOLA1IAPPCES1
SCHEMBL11099793 0.88 TRPA1 (0.60) TRPA1POLBPOLA1IAPPCES1
SCHEMBL22133139 0.86 IAPP (0.43) TRPA1POLBPOLA1IAPPCES1
SCHEMBL2542739 0.86 IAPP (0.43) TRPA1POLBPOLA1IAPPCES1
SCHEMBL11129864 0.80 FAAH (0.64) TRPA1POLBPOLA1CES1CES2
SCHEMBL11129860 0.80 FAAH (0.64) TRPA1POLBPOLA1CES1CES2
SCHEMBL29639616 0.79 TRPA1 (0.63) TRPA1POLBPOLA1CES1CES2
SCHEMBL2081591 0.79 TRPA1 (0.52) TRPA1POLBPOLA1IAPPCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945606-A1 ALKYLCARBAMOYL NAPHTHALENYLOXY- OCTENOYLHYDROXYAMIDE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND PREPARATION THEREOF Korea Research Institute of Chemical Technology (KR) 2008-07-23 EP claimed
WO-2007052938-A1 ALKYLCARBAMOYL NAPHTHALENYLOXY- OCTENOYLHYDROXYAMIDE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2007-05-10 WO claimed