SCHEMBL5024145

SCHEMBL5024145

CN(C[C@H]1CC[C@H](C(=O)NC2CC2)CC1)c1ncc(Br)cn1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 2/20 0.37
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
DRD2 P14416 4/20 0.35
DRD3 P35462 3/20 0.35
HTR2A P28223 2/20 0.35
MELK Q14680 4/20 0.34
FPR3 P25089 1/20 0.34
FPR2 P25090 1/20 0.34
HTR1A P08908 1/20 0.34
POLB P06746 1/20 0.34
EPHX2 P34913 1/20 0.34
GRIN2B Q13224 1/20 0.34
SMO Q99835 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5024150 1.00 KMT2A (0.40) KMT2AMEN1ALDH1A1PKMNPSR1
SCHEMBL5025673 0.83 TAS2R14 (0.38) KMT2AMEN1ALDH1A1NPSR1POLB
SCHEMBL5025675 0.83 TAS2R14 (0.38) KMT2AMEN1ALDH1A1NPSR1POLB
SCHEMBL20772888 0.81 DAO (0.36) GRIN2B
SCHEMBL6013543 0.75 KMT2A (0.44) KMT2AMEN1ALDH1A1NPSR1DRD2
SCHEMBL5024054 0.74 HTT (0.54) KMT2APOLBGRIN2B
SCHEMBL5024052 0.74 HTT (0.54) KMT2APOLBGRIN2B
SCHEMBL5024111 0.71 PLG (0.35) KMT2AMEN1ALDH1A1DRD2MELK
SCHEMBL5028495 0.71 PLG (0.35) KMT2AMEN1ALDH1A1DRD2MELK
SCHEMBL5025789 0.71 HTT (0.41) KMT2AMEN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442791-B2 Aminoalkylamide substituted cyclohexyl derivatives HOFFMANN-LA ROCHE INC. (US) 2008-10-28 US disclosed
EP-1667962-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-06-14 EP disclosed
WO-2005028427-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-03-31 WO disclosed
US-20050065210-A1 Aminoalkylamide substituted cyclohexyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2005-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065210-A1 Aminoalkylamide substituted cyclohexyl derivatives LSS, CYP51A1, CYP46A1 KMT2A 1378/4885MEN1 989/4885ALDH1A1 2099/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.