SCHEMBL6013543

SCHEMBL6013543

O=C(NC1CC1)[C@H]1CC[C@H](CNCc2ncc(Br)cn2)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 5/20 0.38
HPGD P15428 2/20 0.38
DRD2 P14416 3/20 0.38
NPSR1 Q6W5P4 1/20 0.37
HTR2A P28223 2/20 0.36
DRD3 P35462 2/20 0.36
POLB P06746 1/20 0.36
CYP46A1 Q9Y6A2 1/20 0.35
FPR3 P25089 1/20 0.35
FPR2 P25090 1/20 0.35
NPY5R Q15761 1/20 0.35
CCNK O75909 1/20 0.35
CDK9 P50750 1/20 0.35
EPHX2 P34913 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025670 0.84 KMT2A (0.42) KMT2AMEN1ALDH1A1LMNA
SCHEMBL5024150 0.75 KMT2A (0.40) KMT2AMEN1ALDH1A1DRD2NPSR1
SCHEMBL5024145 0.75 KMT2A (0.40) KMT2AMEN1ALDH1A1DRD2NPSR1
SCHEMBL5024050 0.73 HTT (0.53) KMT2AMEN1ALDH1A1HPGDNPSR1
SCHEMBL5024109 0.73 CHRM4 (0.39) KMT2AMEN1ALDH1A1DRD2POLB
SCHEMBL5025785 0.71 SIGMAR1 (0.38) KMT2AMEN1ALDH1A1HPGDNPSR1
SCHEMBL5025524 0.68 KMT2A (0.43) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL2542380 0.68 SMYD3 (0.48) KMT2AMEN1ALDH1A1HPGD
SCHEMBL103961 0.66
SCHEMBL1292139 0.66 VCP (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667962-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-06-14 EP disclosed
WO-2005028427-A1 AMINOALKYLAMIDE SUBSTITUTED CYCLOHEXYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-03-31 WO disclosed