SCHEMBL5024475

SCHEMBL5024475

Cc1c(F)c(F)cc(-c2cc(CCCN3CCCCC3)nc(C#N)n2)c1F

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 16/20 0.54
KCNH2 Q12809 6/20 0.54
CTSS P25774 8/20 0.54
CTSB P07858 1/20 0.54
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5022259 0.81 CTSK (0.48) CTSKKCNH2CTSSCTSB
SCHEMBL5018049 0.79 CTSK (0.43) CTSKKCNH2CTSSCTSB
SCHEMBL5017262 0.77 CTSK (0.39) CTSKKCNH2CTSSCTSB
SCHEMBL5017270 0.76 CTSK (0.42) CTSKKCNH2CTSSCTSB
SCHEMBL5024453 0.75 CTSK (0.56) CTSKKCNH2CTSSCTSB
SCHEMBL13709388 0.74 CTSK (0.57) CTSKKCNH2CTSSCTSBNOS3
SCHEMBL5017183 0.73 CTSK (0.55) CTSKKCNH2CTSSCTSB
SCHEMBL8269456 0.71 CTSK (1.00) CTSKKCNH2CTSSCTSBHRH3
SCHEMBL4446030 0.70 CTSK (1.00) CTSKKCNH2CTSSCTSB
SCHEMBL4440710 0.70 CTSK (1.00) CTSKKCNH2CTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758870-B1 4-PHENYL-PYRIMIDINE-2-CARBONITRILE DERIVATIVES ORGANON NV (NL) 2008-08-13 EP claimed