SCHEMBL5025626

SCHEMBL5025626

O=C(O)N1CC2CCC(O)C(c3ccccc3)C2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GRIN2B Q13224 1/20 0.37
TSHR P16473 1/20 0.36
ATM Q13315 1/20 0.36
HDAC4 P56524 3/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
EPHX2 P34913 1/20 0.35
SLC18A3 Q16572 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA7 P36544 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2800431 1.00 RAB9A (0.37) RAB9ANPC1TP53SMN1; SMN2GRIN2B
SCHEMBL27648867 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL3177278 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL3184361 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL5989023 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL3172844 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL3181798 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL3180166 0.87 TACR1 (0.44) RAB9ANPC1GRIN2BATMEPHX2
SCHEMBL705741 0.82 HDAC4 (0.39) SMN1; SMN2GRIN2BTSHRHDAC4
SCHEMBL13461072 0.82 GPR119 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1898905-A2 HYDROISOINDOLINE TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2008-03-19 EP disclosed
WO-2007002457-A2 HYDROISOINDOLINE TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2007-01-04 WO disclosed