SCHEMBL5026047

SCHEMBL5026047

NCCC[C@H](NC(=O)C(N)CC(=O)N(CCN)CCN)C(=O)N[C@@H](Cc1ccc(C(F)(F)F)cc1)C(=O)Nc1cnc2ccccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.45
HDAC1 Q13547 4/20 0.42
HDAC4 P56524 3/20 0.42
HDAC3 O15379 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC10 Q969S8 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
BDKRB2 P30411 1/20 0.40
CTNNB1 P35222 2/20 0.39
SCN9A Q15858 1/20 0.38
ADCY6 O43306 1/20 0.38
ADCY3 O60266 1/20 0.38
ADCY9 O60503 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5018473 1.00 MCHR1 (0.45) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018157 0.95 BDKRB2 (0.43) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018144 0.95 BDKRB2 (0.43) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018488 0.95 BDKRB2 (0.43) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5024650 0.91 HDAC1 (0.42) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018284 0.90 BDKRB2 (0.41) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018158 0.89 MCHR1 (0.44) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018101 0.89 MCHR1 (0.44) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL5018179 0.89 MCHR1 (0.44) MCHR1HDAC1HDAC4HDAC3HDAC7
SCHEMBL1245446 0.88 BDKRB2 (0.46) MCHR1HDAC1HDAC4HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178490-B2 Polybasic bacterial efflux pump inhibitors and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2012-05-15 US disclosed