SCHEMBL5024650

SCHEMBL5024650

NCCC[C@H](NC(=O)[C@H](N)CC(=O)N(CCN)CCN)C(=O)N[C@@H](Cc1ccc(OC(F)(F)F)cc1)C(=O)Nc1cnc2ccccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.42
HDAC4 P56524 3/20 0.42
BDKRB2 P30411 1/20 0.42
HDAC3 O15379 2/20 0.41
HDAC7 Q8WUI4 2/20 0.41
HDAC2 Q92769 2/20 0.41
HDAC10 Q969S8 2/20 0.41
HDAC11 Q96DB2 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC9 Q9UKV0 2/20 0.41
HDAC5 Q9UQL6 2/20 0.41
CTNNB1 P35222 9/20 0.39
KLKB1 P03952 1/20 0.39
SCN9A Q15858 1/20 0.38
CDH1 P12830 2/20 0.36
TCF7 P36402 2/20 0.36
TCF4 P15884 1/20 0.36
MCHR1 Q99705 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5018473 0.91 MCHR1 (0.45) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5026047 0.91 MCHR1 (0.45) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5018250 0.90 BDKRB2 (0.44) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL13991994 0.87 BDKRB2 (0.43) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5018144 0.86 BDKRB2 (0.43) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5018488 0.86 BDKRB2 (0.43) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5018157 0.86 BDKRB2 (0.43) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5025439 0.85 TRPV1 (0.45) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL13991926 0.85 SCN9A (0.47) HDAC1HDAC4BDKRB2HDAC3HDAC7
SCHEMBL5018317 0.84 LTA4H (0.44) HDAC1HDAC4BDKRB2HDAC3HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178490-B2 Polybasic bacterial efflux pump inhibitors and therapeutic uses thereof REMPEX PHARMACEUTICALS, INC. (US) 2012-05-15 US disclosed