SCHEMBL5029408

SCHEMBL5029408

O=C(O)Nc1nccc(C(F)(F)F)c1O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 3/20 0.40
DHODH Q02127 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
KMO O15229 3/20 0.36
TRPV1 Q8NER1 2/20 0.35
GRM4 Q14833 2/20 0.34
NR3C2 P08235 2/20 0.34
GRIN3B O60391 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2C Q14957 1/20 0.34
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031603 0.85 NR3C2 (0.44) SORT1DHODHHDAC6NR3C2GRIN3B
SCHEMBL23209358 0.74 DPP4 (0.38) SORT1DHODHKMOSMARCA2SMARCA4
SCHEMBL20839296 0.73 HTT (0.39) SORT1DHODHHDAC6TRPV1
SCHEMBL28026509 0.72 SMARCA2 (0.38) SORT1KMOGRM4SMARCA2SMARCA4
SCHEMBL17700420 0.70 SMN1; SMN2 (0.34) SORT1DHODHHDAC6NR3C2GRIN3B
SCHEMBL9998439 0.68 CNR2 (0.46) SORT1DHODH
SCHEMBL11710154 0.67 NOS3 (0.39) KMO
SCHEMBL28603420 0.66 DHODH (0.40) SORT1DHODHHDAC6KMOGRIN3B
SCHEMBL24598127 0.66 SMN1; SMN2 (0.47)
SCHEMBL1652624 0.66 NPC1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957485-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer Healthcare, LLC (US) 2008-08-20 EP disclosed
WO-2007064931-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC (US) 2007-06-07 WO disclosed