SCHEMBL5031603

SCHEMBL5031603

NC(=O)Nc1nccc(C(F)(F)F)c1O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 8/20 0.44
KIF11 P52732 2/20 0.38
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2C Q14957 1/20 0.36
PEPD P12955 1/20 0.34
DHODH Q02127 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
SORT1 Q99523 1/20 0.34
MAPK3 P27361 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5029408 0.85 SORT1 (0.40) NR3C2GRIN3BGRIN1GRIN2CDHODH
SCHEMBL30948751 0.79 NR3C2 (0.47) NR3C2DHODHHDAC6
SCHEMBL11710154 0.70 NOS3 (0.39)
SCHEMBL2787917 0.67 PEPD (0.39) NR3C2KIF11PEPDALDH1A1
SCHEMBL6907368 0.66 NR3C2 (0.36) NR3C2KIF11PEPDALDH1A1
SCHEMBL30875900 0.66 NR3C2 (0.67) NR3C2KIF11SORT1ALDH1A1
SCHEMBL30595621 0.66 SMARCA2 (0.64) NR3C2KIF11HDAC6
SCHEMBL15992647 0.66 SMARCA2 (0.64) NR3C2KIF11HDAC6
SCHEMBL5029590 0.66 NR3C2 (0.67) NR3C2KIF11SORT1ALDH1A1
SCHEMBL24598127 0.65 SMN1; SMN2 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957485-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS Bayer Healthcare, LLC (US) 2008-08-20 EP claimed
WO-2007064931-A2 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC (US) 2007-06-07 WO claimed