SCHEMBL5030195

SCHEMBL5030195

COc1c(F)cccc1C#N.COc1c(F)cccc1C(=N)N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.38
F10 P00742 2/20 0.37
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
HTR2A P28223 1/20 0.34
HCRTR2 O43614 4/20 0.34
HCRTR1 O43613 2/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
SLC6A3 Q01959 1/20 0.33
KLK1 P06870 1/20 0.33
KLK5 Q9Y337 1/20 0.33
TSHR P16473 2/20 0.33
ALDH1A1 P00352 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KAT6A Q92794 1/20 0.32
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135906 0.87 F10 (0.41) F10PRSS1PRSS2PRSS3HCRTR2
SCHEMBL679158 0.83 AR (0.47) ARHTR2AJAK1TYK2SLC6A3
SCHEMBL19638974 0.78 AR (0.41) ARHTR2AHCRTR2HCRTR1JAK1
Hydrochloric Acid SCHEMBL28326198 0.74 IRAK4 (0.36) F10PRSS1PRSS2PRSS3HCRTR2
Hydrochloric Acid SCHEMBL28517935 0.71 F2 (0.43) F10
SCHEMBL6736896 0.71 POLB (0.47) ARTSHRALDH1A1POLBGAA
SCHEMBL16950829 0.71 ALDH1A1 (0.39) JAK1TYK2TSHRALDH1A1NPC1
SCHEMBL528652 0.71 LMNA (0.43) JAK1TYK2TSHRALDH1A1NPC1
SCHEMBL28613887 0.70 KMT2A (0.39) ARALDH1A1KAT6APOLBGAA
SCHEMBL11229875 0.69 TSHR (0.41) F10PRSS1PRSS2PRSS3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951244-A2 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP disclosed
WO-2007062370-A2 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO disclosed