SCHEMBL5030210

SCHEMBL5030210

CCc1cnc(N(C)CC2CCC(NC3CC3)(C(=O)O)CC2)nc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.34
ACACB O00763 3/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
CDK12 Q9NYV4 1/20 0.32
DYRK1A Q13627 1/20 0.30
HCAR3 P49019 1/20 0.30
GPR132 Q9UNW8 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
MELK Q14680 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5025534 0.76 TAS2R14 (0.40) GRIN2BACACB
SCHEMBL5025529 0.76 TAS2R14 (0.40) GRIN2BACACB
SCHEMBL5030212 0.72 TAS2R14 (0.38) GRIN2B
SCHEMBL5028491 0.69 GRIN2B (0.35) GRIN2BACACB
SCHEMBL5762331 0.66 GRIN2B (0.32) GRIN2BACACB
SCHEMBL5762324 0.66 GRIN2B (0.32) GRIN2BACACB
SCHEMBL5028487 0.66 GRIN2B (0.35) GRIN2BACACBCDK12
SCHEMBL12503235 0.65 ALDH1A1 (0.39) ACACBHCAR3
SCHEMBL5026543 0.65 TAS2R14 (0.35)
SCHEMBL5026538 0.65 TAS2R14 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442791-B2 Aminoalkylamide substituted cyclohexyl derivatives HOFFMANN-LA ROCHE INC. (US) 2008-10-28 US disclosed