SCHEMBL28347463

SCHEMBL28347463

NC(=O)Oc1ccccc1NC(=O)c1ccc(C=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
AHR P35869 2/20 0.53
NPC1 O15118 1/20 0.53
NR1I2 O75469 1/20 0.53
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
RAB9A P51151 1/20 0.53
TAAR1 Q96RJ0 1/20 0.53
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 3/20 0.46
GAA P10253 1/20 0.46
MLYCD O95822 1/20 0.45
HPGD P15428 1/20 0.44
F10 P00742 1/20 0.43
PABPC1 P11940 1/20 0.43
APOBEC3A P31941 1/20 0.43
EIF4H Q15056 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
PDCD1 Q15116 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30091844 0.85 NPC1 (0.57) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL22640298 0.83 MLYCD (0.64) KMT2AAHRNPC1RAB9AMEN1
SCHEMBL28901074 0.81 KMT2A (0.57) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL28010642 0.80 KMT2A (0.47) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL12506316 0.80 CACNA1B (0.57) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL28254575 0.80 KMT2A (0.56) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL4887544 0.79 HDAC1 (0.49) KMT2AAHRNPC1NR1I2LMNA
Hydrochloric Acid SCHEMBL28346870 0.79 HDAC2 (0.44) KMT2AAHRNPC1NR1I2LMNA
SCHEMBL8349329 0.78 HDAC1 (0.70) NPC1RAB9AHDAC1HDAC3HDAC2
SCHEMBL3726558 0.77 ALDH1A1 (0.53) KMT2AAHRNPC1NR1I2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111848454-B Histone deacetylase 6 inhibitor and preparation method and application thereof 山东大学 2021-05-07 CN disclosed
CN-111848454-A Histone deacetylase 6 inhibitor and preparation method and application thereof 山东大学 2020-10-30 CN disclosed
CN-110573497-A Histone deacetylase inhibitors 生物马林药物股份有限公司 2019-12-13 CN disclosed