SCHEMBL5031297

SCHEMBL5031297

N#Cc1ccc(NC2CCNC2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
IDO1 P14902 1/20 0.42
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
AXL P30530 5/20 0.40
SLC22A12 Q96S37 3/20 0.39
TRPV4 Q9HBA0 1/20 0.38
P2RX7 Q99572 1/20 0.38
CHEK1 O14757 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3022620 1.00 DPP4 (0.47) DPP4HDAC8HDAC6IDO1NOS3
SCHEMBL9984392 0.92 HDAC8 (0.48) DPP4HDAC8HDAC6IDO1NOS3
Hydrochloric Acid SCHEMBL382423 0.90 HDAC8 (0.47) DPP4HDAC8HDAC6IDO1NOS3
SCHEMBL21460294 0.82 SLC6A2 (0.44) AXLP2RX7
SCHEMBL12596703 0.77 PRKCI (0.44) DPP4AXLCHEK1
SCHEMBL3125940 0.77 HDAC8 (0.48) DPP4HDAC8HDAC6IDO1SLC22A12
SCHEMBL25905013 0.77 HDAC8 (0.48) DPP4HDAC8HDAC6IDO1SLC22A12
Hydrochloric Acid SCHEMBL1032875 0.76 PRKCI (0.43) DPP4AXLCHEK1
Hydrochloric Acid SCHEMBL1032874 0.76 PRKCI (0.43) DPP4AXLCHEK1
SCHEMBL21460253 0.75 DRD2 (0.49) IDO1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954133-A2 PYRROLIDINEANILINES SMITHKLINE BEECHAM CORPORATION (US) 2008-08-13 EP disclosed
WO-2007065093-A2 PYRROLIDINEANILINES SMITHKLINE BEECHAM CORPORATION (US) 2007-06-07 WO disclosed