SCHEMBL5031978

SCHEMBL5031978

COc1ccccc1-c1nc2c(c(=O)[nH]1)CCCC2.COc1ccccc1-c1nc2c(c(=O)n1CCc1ccccc1Cl)CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 6/20 0.44
TNKS2 Q9H2K2 6/20 0.44
HPGD P15428 6/20 0.44
LMNA P02545 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TSHR P16473 2/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PARP10 Q53GL7 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
MAPK1 P28482 1/20 0.42
TNF P01375 1/20 0.41
NOD2 Q9HC29 1/20 0.41
NOD1 Q9Y239 1/20 0.41
PDE5A O76074 1/20 0.37
PARP1 P09874 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4140425 0.91 LMNA (0.42) TNKSTNKS2HPGDLMNAMEN1
SCHEMBL4148644 0.79 KDM4E (0.66) TNKSTNKS2HPGDTSHRKDM4E
SCHEMBL4142349 0.78 TP53 (0.51) TNKSTNKS2KMT2AALDH1A1HTT
SCHEMBL4147903 0.78 CASR (0.47) HPGDLMNAMEN1KMT2ATSHR
SCHEMBL10150419 0.77 KDM4E (0.62) TNKSTNKS2HPGDTSHRKDM4E
SCHEMBL4144693 0.72 TNKS (0.42) TNKSTNKS2HPGDLMNATSHR
SCHEMBL4143059 0.71 TP53 (0.49) KMT2AALDH1A1HSD17B10NPSR1
SCHEMBL13851592 0.69 TP53 (0.50) TSHRALDH1A1NPSR1
SCHEMBL4143019 0.69 TP53 (0.49) LMNAMEN1KMT2ATSHRALDH1A1
SCHEMBL4144206 0.68 TP53 (0.51) TNKSTNKS2KMT2AALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951244-A2 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2008-08-06 EP disclosed
WO-2007062370-A2 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-31 WO disclosed