SCHEMBL5031985

SCHEMBL5031985

NC(=O)C(C(=O)N(c1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1)c1ccc(C(=O)Nc2ccccc2N)cc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.59
HDAC1 Q13547 12/20 0.56
HDAC3 O15379 1/20 0.49
HDAC2 Q92769 1/20 0.49
RXFP1 Q9HBX9 6/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031042 0.85 HDAC1 (0.71) PTGS1HDAC1HDAC3HDAC2
SCHEMBL5126808 0.84 PTGS1 (0.56) PTGS1HDAC1HDAC3HDAC2RXFP1
SCHEMBL5031007 0.82 HDAC1 (0.66) HDAC1HDAC3HDAC2
SCHEMBL5035397 0.81 HDAC1 (0.65) PTGS1HDAC1HDAC3HDAC2
SCHEMBL2107769 0.80 HDAC1 (0.75) PTGS1HDAC1HDAC3HDAC2RXFP1
SCHEMBL5028860 0.77 PTGS1 (0.53) PTGS1HDAC1HDAC3HDAC2
SCHEMBL1689465 0.77 HDAC1 (0.74) PTGS1HDAC1HDAC3HDAC2
SCHEMBL5031052 0.77 HDAC1 (0.60) HDAC1HDAC3HDAC2
SCHEMBL1689312 0.76 HDAC2 (0.62) HDAC1HDAC3HDAC2
SCHEMBL5028824 0.76 HDAC1 (0.56) HDAC1HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed