SCHEMBL5035397

SCHEMBL5035397

NC(=O)C(C(=O)N(c1ccc(F)cc1)c1ccc(F)cc1)c1ccc(C(=O)Nc2ccccc2N)cc1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.65
HDAC2 Q92769 7/20 0.55
HDAC3 O15379 6/20 0.55
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
PTGS1 P23219 1/20 0.49
MAPK1 P28482 1/20 0.49
NCOR2 Q9Y618 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5031042 0.91 HDAC1 (0.71) HDAC1HDAC2HDAC3PTGS1MAPK1
SCHEMBL1689343 0.86 HDAC1 (0.54) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL1689164 0.82 HDAC1 (0.60) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL5031015 0.82 HDAC1 (0.70) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL5031985 0.81 PTGS1 (0.59) HDAC1HDAC2HDAC3PTGS1
SCHEMBL1689344 0.81 HDAC1 (0.53) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL28188848 0.80 MEN1 (0.77) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL5031007 0.79 HDAC1 (0.66) HDAC1HDAC2HDAC3MEN1KMT2A
SCHEMBL5031052 0.79 HDAC1 (0.60) HDAC1HDAC2HDAC3
SCHEMBL2109945 0.79 HDAC1 (1.00) HDAC1HDAC2HDAC3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP disclosed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO disclosed