SCHEMBL5033456

SCHEMBL5033456

C=CC(=S)N1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.50
CA1 P00915 3/20 0.50
CA9 Q16790 3/20 0.50
CA2 P00918 2/20 0.50
MAPT P10636 2/20 0.50
MGLL Q99685 6/20 0.48
ALDH1A1 P00352 6/20 0.48
PDK1 Q15118 2/20 0.48
PDK2 Q15119 2/20 0.48
PDK3 Q15120 2/20 0.48
PHGDH O43175 2/20 0.48
FAAH O00519 1/20 0.48
ALDH2 P05091 1/20 0.48
KDM4E B2RXH2 3/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TSHR P16473 1/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
AGTR1 P30556 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28820714 0.77
SCHEMBL24517883 0.75 CA1 (0.46) CA12CA1CA9CA2MAPT
SCHEMBL15154762 0.73 MAPT (0.42) CA12CA1CA9CA2MAPT
SCHEMBL19566767 0.73 MAPT (0.42) CA12CA1CA9CA2MAPT
SCHEMBL16178713 0.71 SMN1; SMN2 (0.48) CA12CA1CA9CA2MAPT
SCHEMBL20547256 0.71 MEN1 (0.52) CA12CA1CA9MAPTALDH1A1
SCHEMBL19245083 0.71 LMNA (0.43) CA12CA1CA9CA2MAPT
SCHEMBL36422 0.71 MEN1 (0.52) CA12CA1CA9MAPTALDH1A1
SCHEMBL20253609 0.71 MAPT (0.55) CA12CA1CA9CA2MAPT
SCHEMBL17934675 0.70 MAPT (0.44) CA12CA1CA9CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007393-A2 THIAZOLE AND THIOPHENE ANALOGUES, AND THEIR USE IN TREATING AUTOIMMUNE DISEASES AND CANCERS Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College (US) 2008-12-31 EP disclosed
WO-2007118149-A2 THIAZOLE AND THIOPHENE ANALOGUES, AND THEIR USE IN TREATING AUTOIMMUNE DISEASES AND CANCERS BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL LOLLEGE (US) 2007-10-18 WO disclosed