SCHEMBL5034006

SCHEMBL5034006

CCCC[P+](CCCC)(CCCC)CCCC.[C-]#N

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DNM1 Q05193 2/20 0.67
BDKRB2 P30411 2/20 0.39
TSHR P16473 5/20 0.38
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
CYP3A4 P08684 1/20 0.36
FDPS P14324 1/20 0.36
THRB P10828 1/20 0.35
OPRM1 P35372 1/20 0.35
CA2 P00918 2/20 0.35
MAPK1 P28482 1/20 0.35
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29496398 0.89 DNM1 (0.80) DNM1BDKRB2TSHRALDH1A1TDP1
Bromide SCHEMBL126636 0.86 DNM1 (0.81) DNM1BDKRB2TSHRALDH1A1TDP1
Phosphine SCHEMBL31655327 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
SCHEMBL30703682 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
Bromide SCHEMBL302420 0.86 DNM1 (0.81) DNM1BDKRB2TSHRALDH1A1TDP1
Hydrochloric Acid SCHEMBL23198627 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
SCHEMBL9303471 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
Hydrochloric Acid SCHEMBL124627 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
Iodide SCHEMBL187956 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1
SCHEMBL29769886 0.86 DNM1 (0.75) DNM1BDKRB2TSHRALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005375-A1 METHOD FOR PRODUCING 4-CYANO-3-HYDROXYBUTYRIC ACID ESTERS LANXESS DEUTSCHLAND GMBH (DE) 2005-01-20 WO claimed
WO-1995001962-A1 PROCESS FOR THE PREPARATION OF CHIRAL 3-(1-AMINO-1,1-BISALKYLMETHYL)-1-SUBSTITUTED-PYRROLIDINES WARNER-LAMBERT COMPANY (US) 1995-01-19 WO claimed
US-5347017-A Process for chiral 3-(1-amino-1,1-bisalkylmethyl)-1-substituted-pyrrolidines WARNER-LAMBERT COMPANY (US) 1994-09-13 US claimed
EP-3604276-A1 NEW COMPONENTS FOR ELECTROLYTE COMPOSITIONS SOLVAY SA (BE) 2020-02-05 EP disclosed
US-7423162-B2 Process for the preparation of (4-hydroxy-6-oxo-tetrahydropyran-2-yl) acetonitrile and derivatives DSM IP ASSETS B.V. (NL) 2008-09-09 US disclosed
EP-1620423-B1 PROCESS FOR THE PREPARATION OF (4-HYDROXY-6-OXO-TETRAHYDROPYRAN-2-YL) ACETONITRILE AND DERIVATIVES THEREOF DSM IP ASSETS BV (NL) 2008-02-20 EP disclosed
WO-2007137816-A1 PROCESS FOR THE PREPARATION OF EPOXIDE INTERMEDIATES FOR PHARMACEUTICAL COMPOUNDS SUCH AS STATINS DSM IP ASSETS B.V. (NL) 2007-12-06 WO disclosed
WO-2007128469-A1 PROCESS FOR THE PREPARATION OF ENANTIOMERICALLY ENRICHED NITRILES DSM IP ASSETS B.V. (NL) 2007-11-15 WO disclosed
US-20060258733-A1 By reacting 2-(leaving group-methyl)-4-hydroxy-6-oxotetrahydropyran with a cyanide ion in water at a pH of 0-5; nitrile may be reduced to form an aminoethyl group; reacting with an acetal-forming agent to form a 1,3-dioxane derivative; may be further converted to atorvastatin or its calcium salt DSM SINOCHEM PHARMACEUTICALS NETHERLANDS B.V. (NL) 2006-11-16 US disclosed
EP-1620423-A1 PROCESS FOR THE PREPARATION OF (4-HYDROXY-6-OXO-TETRAHYDROPYRAN-2-YL) ACETONITRILE AND DERIVATIVES THEREOF DSM IP Assets B.V. (NL) 2006-02-01 EP disclosed
WO-2005005375-A1 METHOD FOR PRODUCING 4-CYANO-3-HYDROXYBUTYRIC ACID ESTERS LANXESS DEUTSCHLAND GMBH (DE) 2005-01-20 WO disclosed
WO-2004096788-A1 PROCESS FOT THE PREPARATION OF (4-HYDROXY-6-OXO-TETRAHYDROPYRAN-2-YL) ACETONITRILE AND DERIVATIVES THEREOF DSM IP ASSETS B.V. (NL) 2004-11-11 WO disclosed
US-5466828-A Chiral 3-cyano-1-substituted-pyrrolidines WARNER-LAMBERT COMPANY (US) 1995-11-14 US disclosed
WO-1995001962-A1 PROCESS FOR THE PREPARATION OF CHIRAL 3-(1-AMINO-1,1-BISALKYLMETHYL)-1-SUBSTITUTED-PYRROLIDINES WARNER-LAMBERT COMPANY (US) 1995-01-19 WO disclosed
US-5347017-A Process for chiral 3-(1-amino-1,1-bisalkylmethyl)-1-substituted-pyrrolidines WARNER-LAMBERT COMPANY (US) 1994-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060258733-A1 By reacting 2-(leaving group-methyl)-4-hydroxy-6-oxotetrahydropyran with a cyanide ion in water at a pH of 0-5; nitrile may be reduced to form an aminoethyl group; reacting with an acetal-forming agent to form a 1,3-dioxane derivative; may be further converted to atorvastatin or its calcium salt HMGCR, CYP11B2, CYP4F2 DNM1 421/4885BDKRB2 3884/4885TSHR 4782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.