SCHEMBL5035176

SCHEMBL5035176

Cc1cc(COc2ccc(-c3cc(CC4(C)NC(=O)NC4=O)no3)cc2)c2ccccc2n1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 8/20 0.60
MMP13 P45452 1/20 0.58
MMP2 P08253 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5032791 0.94 ADAM17 (0.58) ADAM17MMP13
SCHEMBL5032796 0.78 ADAM17 (0.46) ADAM17MMP13MMP2
SCHEMBL5032806 0.77 MMP13 (0.51) ADAM17MMP13MMP2
SCHEMBL4050333 0.77 ADAM17 (0.76) ADAM17MMP13MMP2
SCHEMBL6210129 0.76 ADAM17 (0.64) ADAM17MMP13MMP2
SCHEMBL6321457 0.76 ADAM17 (0.74) ADAM17MMP13MMP2
SCHEMBL6210103 0.76 ADAM17 (0.73) ADAM17MMP13MMP2
SCHEMBL4051714 0.76 ADAM17 (0.71) ADAM17MMP13MMP2
SCHEMBL4059418 0.75 ADAM17 (1.00) ADAM17MMP13MMP2
SCHEMBL6210085 0.75 ADAM17 (0.70) ADAM17MMP13MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628974-A4 HYDANTOIN DERIVATIVES AS INHIBITORS OF TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME (TACE) BRISTOL MYERS SQUIBB CO (US) 2008-05-07 EP claimed
EP-1628974-A2 HYDANTOIN DERIVATIVES AS INHIBITORS OF TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME (TACE) Bristol-Myers Squibb Company (US) 2006-03-01 EP claimed
WO-2004108086-A2 HYDANTOIN DERIVATIVES AS INHIBITORS OF TUMOR NECROSIS FACTOR-α CONVERTING ENZYME (TACE) BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-16 WO claimed