SCHEMBL5035185

SCHEMBL5035185

CN1C=CC(N(C)c2nc(Nc3ccc(OCOP(=O)(O)O)c(F)c3)nc(NC3CCCCCC3)n2)CC1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.38
CCNT1 O60563 1/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCND3 P30281 1/20 0.37
CDK9 P50750 1/20 0.37
CDK6 Q00534 1/20 0.37
AXL P30530 8/20 0.36
BCL6 P41182 2/20 0.35
SIK1 P57059 1/20 0.34
SIK2 Q9H0K1 1/20 0.34
SIK3 Q9Y2K2 1/20 0.34
MAPK8 P45983 2/20 0.34
IDH2 P48735 1/20 0.33
INSR P06213 1/20 0.33
ALK Q9UM73 1/20 0.33
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4838644 0.88 IDH2 (0.40) EGFRCCNT1CDK4CCND1CCND3
SCHEMBL5032511 0.82 RAB9A (0.39) IDH2
SCHEMBL5032373 0.80 SMN1; SMN2 (0.39) BCL6MAPK8
SCHEMBL14268424 0.80 EGFR (0.40) EGFRAXLBCL6
SCHEMBL4870097 0.79 BCL6 (0.42) EGFRCCND3CDK6AXLBCL6
SCHEMBL4837995 0.79 IDH2 (0.42) EGFRAXLBCL6SIK1SIK2
SCHEMBL5032431 0.78 NPSR1 (0.38) CDK4CCND1BCL6
SCHEMBL4832236 0.78 IDH2 (0.43) EGFRCCNT1CDK4CCND1CCND3
SCHEMBL4836907 0.77 GALR1 (0.40) EGFRAXLBCL6
SCHEMBL4832431 0.76 IDH2 (0.44) EGFRCCNT1CDK4CCND1CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7335656-B2 Stent with a disposed traiazine compound such as 6-(3-Chloro-4-methoxy-phenoxy)-N-cycloheptyl-N'-methyl-N'-(1-methyl-piperidin-4-yl)-[1,3,5]triazine-2,4-diamine for inhibiting smooth muscle proliferation; restenosis and atherosclerosis REDDY US THERAPEUTICS, INC. (US) 2008-02-26 US disclosed