SCHEMBL5035270

SCHEMBL5035270

NS(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C(F)F)cc(-c4ccc(Cl)cc4)nc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.54
KMT2A Q03164 3/20 0.53
KDM4E B2RXH2 3/20 0.53
HTT P42858 1/20 0.53
CA2 P00918 8/20 0.47
CA1 P00915 7/20 0.47
CA9 Q16790 6/20 0.47
CA12 O43570 5/20 0.47
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
TP53 P04637 4/20 0.46
POLB P06746 2/20 0.46
THRB P10828 1/20 0.44
MAPT P10636 3/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CA4 P22748 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034903 0.92 MAPK1 (0.52) MAPK1KMT2AKDM4EHTTCA2
SCHEMBL5034992 0.91 MAPK1 (0.52) MAPK1KMT2AKDM4EHTTCA2
SCHEMBL5034977 0.90 KDM4E (0.52) MAPK1KMT2AKDM4EHTTCA2
SCHEMBL5034984 0.89 KDM4E (0.54) MAPK1KMT2AKDM4EHTTCA2
SCHEMBL5036051 0.89 MAPK1 (0.49) MAPK1KMT2AKDM4EHTTCA2
SCHEMBL5032671 0.88 MAPK1 (0.71) MAPK1KMT2AKDM4EHTTALDH1A1
SCHEMBL5036107 0.88 MAPK1 (0.52) MAPK1KMT2AKDM4EHTTALDH1A1
SCHEMBL5041510 0.88 CA2 (0.52) KMT2AKDM4EHTTCA2CA1
SCHEMBL5039198 0.87 CA2 (0.48) MAPK1KMT2AKDM4ECA2CA1
SCHEMBL5041958 0.87 MAPK1 (0.65) MAPK1KMT2AKDM4EHTTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed