SCHEMBL5035278

SCHEMBL5035278

Cc1cc(-c2ccc(C(F)(F)F)cc2)nc2c(OC(=O)Nc3cccc(S(N)(=O)=O)c3)cnn12

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.44
CA9 Q16790 4/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.44
CA4 P22748 1/20 0.42
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032666 0.93 NTRK1 (0.44) KDM4EHTTKMT2A
SCHEMBL5039162 0.91 CA12 (0.47) CA2CA9CA12CA1KDM4E
SCHEMBL5041510 0.89 CA2 (0.52) CA2CA9CA12CA1CA4
SCHEMBL5034992 0.89 MAPK1 (0.52) CA2CA9CA12CA1KDM4E
SCHEMBL5036088 0.88 CA12 (0.42) CA2CA9CA12CA1CA4
SCHEMBL5048263 0.86 CA12 (0.53) CA2CA9CA12CA1KDM4E
SCHEMBL5035282 0.85 CA2 (0.46) CA2CA9CA12CA1
SCHEMBL5035013 0.85 KDM4E (0.46) KDM4EHTTKMT2A
SCHEMBL5039198 0.84 CA2 (0.48) CA2CA9CA12CA1KDM4E
SCHEMBL5034981 0.83 KDM4E (0.45) KDM4EHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed