SCHEMBL5036059

SCHEMBL5036059

CCOc1cc(-c2cc(C(F)F)n3ncc(OC(=O)Nc4cccc(S(C)(=O)=O)c4)c3n2)ccc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
KMT2A Q03164 3/20 0.47
HTT P42858 1/20 0.47
MAPT P10636 3/20 0.47
MAPK1 P28482 1/20 0.46
TP53 P04637 2/20 0.40
POLB P06746 1/20 0.40
ALDH1A1 P00352 4/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 1/20 0.38
RXFP1 Q9HBX9 2/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034925 0.95 KDM4E (0.48) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5032681 0.94 KDM4E (0.47) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5036085 0.91 THRB (0.44) KDM4EKMT2AHTTMAPTPOLB
SCHEMBL5036170 0.90 KDM4E (0.44) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5041389 0.90 KDM4E (0.46) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5045539 0.90 MAPT (0.58) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5035331 0.90 KDM4E (0.49) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5039093 0.90 KDM4E (0.49) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5036036 0.89 KDM4E (0.51) KDM4EKMT2AHTTMAPTMAPK1
SCHEMBL5041451 0.88 MAPK1 (0.47) KDM4EKMT2AHTTMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed