SCHEMBL5036557

SCHEMBL5036557

CS(=O)(=O)c1cccc(NC(=O)Oc2cnn3c(C4CC4)cc(-c4ccc(Cl)cc4)nc23)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.41
RIPK2 O43353 2/20 0.40
PSD A5PKW4 3/20 0.40
MAPK1 P28482 1/20 0.40
NTRK1 P04629 1/20 0.39
MET P08581 1/20 0.39
PIM1 P11309 1/20 0.39
FGFR1 P11362 1/20 0.39
MAP2K2 P36507 1/20 0.39
FLT3 P36888 1/20 0.39
MAPK8 P45983 1/20 0.39
GSK3B P49841 1/20 0.39
NTRK3 Q16288 1/20 0.39
ALK Q9UM73 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 3/20 0.39
KIF18A Q8NI77 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039328 0.92 CA2 (0.46) KMT2AKDM4EHTTMAPK1CA2
SCHEMBL5035007 0.91 NTRK1 (0.41) KMT2AKDM4EHTTMAPK1NTRK1
SCHEMBL5039084 0.90 KIF18A (0.44) KMT2AKDM4EHTTMAPK1CA2
SCHEMBL5034946 0.90 RIPK2 (0.43) KMT2AKDM4EHTTRIPK2PSD
SCHEMBL5039369 0.88 CA2 (0.43) KMT2AKDM4EHTTRIPK2PSD
SCHEMBL5041408 0.87 KIF18A (0.45) KMT2AKDM4EHTTKIF18A
SCHEMBL5036499 0.87 KMT2A (0.44) KMT2AKDM4EHTTRIPK2PSD
SCHEMBL5039326 0.86 KMT2A (0.40) KMT2AKDM4EHTTRIPK2PSD
SCHEMBL5048443 0.86 MAPK1 (0.50) KMT2AKDM4EHTTRIPK2PSD
SCHEMBL5041442 0.85 KDM4E (0.45) KMT2AKDM4EHTTMAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed