SCHEMBL5037822

SCHEMBL5037822

N#Cc1ccc(OCC2CC2)c(C(=O)N2CCN(c3ccc(C(F)(F)F)cc3)CC2)c1

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 17/20 0.71
KCNH2 Q12809 5/20 0.58
CETP P11597 1/20 0.43
CA12 O43570 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041864 0.89 SLC6A9 (0.60) SLC6A9KCNH2CETPCA12CA2
SCHEMBL5042735 0.86 SLC6A9 (0.56) SLC6A9KCNH2CETP
SCHEMBL5041322 0.86 SLC6A9 (0.59) SLC6A9KCNH2CETP
SCHEMBL5047602 0.85 SLC6A9 (0.58) SLC6A9KCNH2CETPCA12CA2
SCHEMBL4426863 0.83 SLC6A9 (0.72) SLC6A9KCNH2
SCHEMBL4433387 0.83 SLC6A9 (1.00) SLC6A9KCNH2
SCHEMBL4425004 0.83 SLC6A9 (0.70) SLC6A9KCNH2CETP
SCHEMBL4421782 0.81 SLC6A9 (0.82) SLC6A9KCNH2
SCHEMBL4427060 0.80 SLC6A9 (0.77) SLC6A9KCNH2
SCHEMBL4419780 0.80 SLC6A9 (0.93) SLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed