SCHEMBL5041864

SCHEMBL5041864

N#Cc1ccc(OCC(F)(F)F)c(C(=O)N2CCN(c3ccc(C(F)(F)F)cc3)CC2)c1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 15/20 0.60
KCNH2 Q12809 5/20 0.60
CETP P11597 1/20 0.45
CA12 O43570 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
ENPP2 Q13822 2/20 0.43
AKR1C3 P42330 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037822 0.89 SLC6A9 (0.71) SLC6A9KCNH2CETPCA12CA2
SCHEMBL5041322 0.89 SLC6A9 (0.59) SLC6A9KCNH2CETP
SCHEMBL5042735 0.89 SLC6A9 (0.56) SLC6A9KCNH2CETP
SCHEMBL4425004 0.85 SLC6A9 (0.70) SLC6A9KCNH2CETP
SCHEMBL5047534 0.84 SLC6A9 (0.78) SLC6A9KCNH2
SCHEMBL5047602 0.83 SLC6A9 (0.58) SLC6A9KCNH2CETPCA12CA2
SCHEMBL5042095 0.82 SLC6A9 (0.65) SLC6A9KCNH2
SCHEMBL4427344 0.81 SLC6A9 (0.66) SLC6A9KCNH2ENPP2
SCHEMBL4425925 0.79 SLC6A9 (0.65) SLC6A9KCNH2
SCHEMBL4908289 0.77 SLC6A9 (0.49) SLC6A9KCNH2CETPCA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed