SCHEMBL5038429

SCHEMBL5038429

N#Cc1ccc(F)cc1Cc1nc(Cl)[nH]c(=O)c1F

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 5/20 0.38
PRMT5 O14744 2/20 0.37
WDR77 Q9BQA1 2/20 0.37
DPP4 P27487 6/20 0.36
MPO P05164 1/20 0.36
DAO P14920 1/20 0.34
HSD11B1 P28845 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502305 0.90 RIPK3 (0.36) IDH1PRMT5WDR77HSD11B1
SCHEMBL6507892 0.89 DPP4 (0.38) IDH1PRMT5WDR77DPP4MPO
SCHEMBL6511158 0.68 DPP4 (0.56) DPP4
SCHEMBL16824548 0.66 MAOA (0.41) IDH1DPP4MPO
SCHEMBL28286565 0.66 MAOA (0.41) IDH1DPP4MPO
SCHEMBL2591940 0.66 SLC22A12 (0.43) IDH1DPP4MPO
SCHEMBL8665297 0.64 HTT (0.37)
SCHEMBL13142036 0.64 DPP4 (0.46) DPP4
SCHEMBL14039187 0.64 MAOA (0.42) IDH1DPP4MPO
SCHEMBL13041692 0.63 HTR2A (0.47) IDH1MPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016911-A1 4-PYRIMIDONE DERIVATIVES AND THEIR USE AS PEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-02-24 WO claimed
EP-1911754-A1 Dipeptidyl peptidase inhibitors Takeda Pharmaceutical Company Limited (JP) 2008-04-16 EP disclosed
WO-2005016911-A1 4-PYRIMIDONE DERIVATIVES AND THEIR USE AS PEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-02-24 WO disclosed