SCHEMBL6507892

SCHEMBL6507892

N#Cc1ccc(F)cc1Cc1nc(Cl)[nH]c(=O)c1Br

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.38
IDH1 O75874 5/20 0.37
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
MPO P05164 1/20 0.35
HSD11B1 P28845 3/20 0.33
DAO P14920 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5038429 0.89 IDH1 (0.38) DPP4IDH1PRMT5WDR77MPO
SCHEMBL6502305 0.80 RIPK3 (0.36) IDH1PRMT5WDR77HSD11B1
SCHEMBL6507784 0.74 DPP4 (0.59) DPP4
SCHEMBL5132430 0.73 PARP1 (0.37) DPP4
SCHEMBL6511158 0.67 DPP4 (0.56) DPP4
SCHEMBL305457 0.65 MAOA (0.41) DPP4IDH1MPO
SCHEMBL16824548 0.65 MAOA (0.41) DPP4IDH1MPO
SCHEMBL28286565 0.65 MAOA (0.41) DPP4IDH1MPO
SCHEMBL2591940 0.65 SLC22A12 (0.43) DPP4IDH1MPO
SCHEMBL3393525 0.64 DPP4 (0.60) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016911-A1 4-PYRIMIDONE DERIVATIVES AND THEIR USE AS PEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-02-24 WO claimed
EP-1911754-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL (JP) 2013-10-09 EP disclosed
WO-2005016911-A1 4-PYRIMIDONE DERIVATIVES AND THEIR USE AS PEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-02-24 WO disclosed