SCHEMBL5041286

SCHEMBL5041286

CCOc1cc(OC2CCN(C)CC2)c(F)c([C@H](OC)C(=O)NCc2ccc(C#N)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.49
HRH3 Q9Y5N1 4/20 0.41
SLC1A2 P43004 2/20 0.40
SLC1A3 P43003 1/20 0.40
HAT1 O14929 2/20 0.39
EP300 Q09472 2/20 0.39
HTR2A P28223 4/20 0.38
KCNH2 Q12809 2/20 0.38
ABCB11 O95342 1/20 0.38
CYP1A2 P05177 1/20 0.38
ADRB2 P07550 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
DRD1 P21728 1/20 0.38
TBXA2R P21731 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2C P28335 1/20 0.38
GPR183 P32249 1/20 0.38
CYP2C19 P33261 1/20 0.38
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5041282 1.00 F10 (0.49) F10HRH3SLC1A2SLC1A3HAT1
SCHEMBL5040925 0.92 F10 (0.43) F10SLC1A2SLC1A3GPR6EPHX2
SCHEMBL5045642 0.90 F10 (0.39) F10HTR2A
SCHEMBL5045638 0.90 F10 (0.39) F10HTR2A
SCHEMBL5040944 0.89 GPR119 (0.50) F10HTR2A
SCHEMBL5042471 0.88 KMT2A (0.43) F10
SCHEMBL5042467 0.88 KMT2A (0.43) F10
SCHEMBL5041188 0.86 MEN1 (0.39) EPHX2
SCHEMBL5041195 0.86 MEN1 (0.39) EPHX2
Hydrochloric Acid SCHEMBL5041666 0.86 F10 (0.66) F10HRH3HTR2AKCNH2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
US-7129238-B2 Mandelic acid derivatives HOFFMANN-LA ROCHE INC. (US) 2006-10-31 US disclosed
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
US-20040122057-A1 Novel mandelic acid derivatives HOFFMANN-LA ROCHE INC. 2004-06-24 US disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122057-A1 Novel mandelic acid derivatives F7, F11, F9 F10 8/4885HRH3 352/4885SLC1A2 2127/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.