SCHEMBL5042669

SCHEMBL5042669

COC(C(=O)NCc1ccc(C(=N)N)cc1)c1cc(Br)ccc1F

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 6/20 0.48
ST14 Q9Y5Y6 1/20 0.46
F2 P00734 8/20 0.44
PKM P14618 1/20 0.41
F7 P08709 4/20 0.40
F10 P00742 3/20 0.40
PRSS1 P07477 2/20 0.40
MASP2 O00187 1/20 0.40
ALDH1A1 P00352 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5042670 1.00 KLKB1 (0.48) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5037655 0.99 KLKB1 (0.47) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5037650 0.99 KLKB1 (0.47) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5047306 0.91 KLKB1 (0.47) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5047303 0.91 KLKB1 (0.47) KLKB1ST14F2PKMF7
SCHEMBL5041859 0.88 PKM (0.49) KLKB1ST14F2PKMF7
SCHEMBL5041852 0.88 PKM (0.49) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5047280 0.88 PKM (0.48) KLKB1ST14F2PKMF7
SCHEMBL5047896 0.88 F2 (0.49) KLKB1ST14F2PKMF7
Hydrochloric Acid SCHEMBL5047289 0.88 PKM (0.48) KLKB1ST14F2PKMF7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-B1 MANDELIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-23 EP disclosed
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed