SCHEMBL5043481

SCHEMBL5043481

CCOc1ccc(S(N)(=O)=O)cc1C(=O)N1CCN(c2ccc(C#N)c(F)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 17/20 0.59
KCNH2 Q12809 6/20 0.49
GAA P10253 1/20 0.47
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424086 0.91 SLC6A9 (0.61) SLC6A9KCNH2GAA
SCHEMBL5042007 0.88 SLC6A9 (0.58) SLC6A9KCNH2GAA
SCHEMBL5043126 0.88 SLC6A9 (0.59) SLC6A9KCNH2GAA
SCHEMBL4425808 0.87 SLC6A9 (0.52) SLC6A9KCNH2GAALMNA
SCHEMBL5043057 0.86 SLC6A9 (0.64) SLC6A9KCNH2GAALMNATSHR
SCHEMBL4424200 0.85 SLC6A9 (0.44) SLC6A9KCNH2GAA
SCHEMBL5038132 0.84 SLC6A9 (0.59) SLC6A9KCNH2GAA
SCHEMBL5042339 0.83 SLC6A9 (0.71) SLC6A9KCNH2
SCHEMBL4423997 0.83 SLC6A9 (0.71) SLC6A9KCNH2
SCHEMBL4424855 0.83 SLC6A9 (0.71) SLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656361-B1 PIPERAZINE WITH OR-SUBSTITUTED PHENYL GROUP AND THEIR USE AS GLYT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed