SCHEMBL5044641

SCHEMBL5044641

COc1ccc2nc(C(C)CN3CC[CH]CC3)c(=O)[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPSR1 Q6W5P4 2/20 0.44
GFER P55789 1/20 0.44
CYP1A2 P05177 7/20 0.43
CYP2E1 P05181 7/20 0.43
CYP3A4 P08684 7/20 0.43
CYP2C8 P10632 7/20 0.43
CYP2D6 P10635 7/20 0.43
CYP2C9 P11712 7/20 0.43
CYP2B6 P20813 7/20 0.43
CYP2C19 P33261 7/20 0.43
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41
KDM4E B2RXH2 2/20 0.41
TP53 P04637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733245 0.78 NPSR1 (0.46) NPC1RAB9ASMN1; SMN2NPSR1GFER
SCHEMBL4308827 0.78 CYP1A2 (0.52) NPC1RAB9ASMN1; SMN2NPSR1GFER
SCHEMBL18557755 0.73 CYP1A2 (0.44) NPC1RAB9ASMN1; SMN2GFERCYP1A2
SCHEMBL620809 0.68 KDM4E (0.55) NPC1RAB9ASMN1; SMN2NPSR1GFER
SCHEMBL4308637 0.68 CYP1A2 (0.52) NPC1RAB9ASMN1; SMN2NPSR1GFER
SCHEMBL4303506 0.68 ALDH1A1 (0.54) NPC1SMN1; SMN2GFERCYP1A2CYP2E1
SCHEMBL29991257 0.68 KDM4E (0.59) NPC1RAB9ASMN1; SMN2CYP1A2CYP2E1
SCHEMBL20595527 0.68 KDM4E (0.59) NPC1RAB9ASMN1; SMN2CYP1A2CYP2E1
SCHEMBL29991190 0.67 NPC1 (0.52) NPC1RAB9ASMN1; SMN2NPSR1GFER
SCHEMBL21800738 0.67 NPC1 (0.52) NPC1RAB9ASMN1; SMN2NPSR1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893599-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS AstraZeneca AB (SE) 2008-03-05 EP disclosed
WO-2006134378-A1 COMPOUNDS FOR THE TREATMENT OF MULTI-DRUG RESISTANT BACTERIAL INFECTIONS ASTRAZENECA AB (SE) 2006-12-21 WO disclosed