SCHEMBL5045201

SCHEMBL5045201

N#Cc1c[nH]c2c(=O)[nH]c(=O)[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPYD Q12882 3/20 0.60
GDA Q9Y2T3 2/20 0.40
MCL1 Q07820 5/20 0.37
DYRK1A Q13627 3/20 0.37
ACHE P22303 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
UPP1 Q16831 1/20 0.32
IMPDH2 P12268 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL189451 0.75 DPYD (1.00) DPYDMCL1KDM4EALDH1A1HPGD
SCHEMBL9008314 0.65 GDA (0.71) DPYDGDAACHEKDM4EALDH1A1
SCHEMBL3254445 0.65 DYRK1A (0.52) DPYDDYRK1AKDM4EALDH1A1IMPDH2
Uric Acid SCHEMBL27548112 0.64 GDA (0.76) DPYDGDAACHEKDM4EALDH1A1
SCHEMBL5048035 0.64 PIM1 (0.40) DPYDGDAACHEKDM4EALDH1A1
SCHEMBL187437 0.64 DPYD (0.64) DPYDMCL1KDM4EALDH1A1HPGD
SCHEMBL3945500 0.63 PNP (0.45) DPYDALDH1A1
Uric Acid SCHEMBL28124016 0.63 GDA (0.73) DPYDGDAACHEKDM4EALDH1A1
Uric Acid SCHEMBL28323281 0.63 GDA (0.73) DPYDGDAACHEKDM4EALDH1A1
Uric Acid SCHEMBL27432318 0.63 GDA (0.73) DPYDGDAACHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966215-A1 CONDENSED HETEROCYCLIC COMPOUNDS USEFUL AS DPP-IV INHIBITORS Novartis AG (CH) 2008-09-10 EP disclosed
WO-2007071738-A1 CONDENSED HETEROCYCLIC COMPOUNDS USEFUL AS DPP-IV INHIBITORS NOVARTIS AG (CH) 2007-06-28 WO disclosed