SCHEMBL5046079

SCHEMBL5046079

N#Cc1cc2c(nc1NCCc1ccccc1)CCCC2=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
KDM4E B2RXH2 2/20 0.60
L3MBTL1 Q9Y468 2/20 0.60
NPSR1 Q6W5P4 2/20 0.60
TSHR P16473 2/20 0.60
MAPT P10636 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
TAAR1 Q96RJ0 1/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
MAPK1 P28482 2/20 0.41
GAA P10253 1/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
TP53 P04637 1/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
NCOA1 Q15788 1/20 0.40
ESR2 Q92731 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035975 0.82 POLB (0.52) ALDH1A1
SCHEMBL8282928 0.80 TSHR (0.57) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4424079 0.80 NPC1 (0.54) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4423396 0.78 ALDH1A1 (0.50) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4433042 0.76 ALDH1A1 (0.52) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4424040 0.75 ALDH1A1 (1.00) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL13673758 0.73 KDM4E (0.60) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4421527 0.73 ALDH1A1 (0.60) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4433628 0.72 ALDH1A1 (0.45) ALDH1A1KDM4EL3MBTL1NPSR1TSHR
SCHEMBL4423371 0.72 ALDH1A1 (0.51) ALDH1A1KDM4EL3MBTL1NPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723116-B1 TETRAHYDROQUINOLINONES AND THEIR USE AS ANTAGONISTS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO KGAA (DE) 2008-09-24 EP claimed