SCHEMBL5046741

SCHEMBL5046741

[N-]=[N+]=C(C(=O)O)c1cccc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.58
NR4A2 P43354 1/20 0.58
NR4A3 Q92570 1/20 0.58
CDC25B P30305 1/20 0.51
MMP3 P08254 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
PTPN1 P18031 1/20 0.47
PLK1 P53350 1/20 0.47
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
HPGD P15428 3/20 0.43
KMT2A Q03164 3/20 0.43
MAPT P10636 3/20 0.43
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346405 0.80 PLK1 (0.50) NR4A1NR4A2NR4A3CDC25BMMP3
SCHEMBL8074423 0.77 CDC25B (0.56) NR4A1NR4A2NR4A3CDC25BPTPN1
SCHEMBL991197 0.76 ERCC5 (0.50) CYP3A4CYP2C9HPGDKMT2AALDH1A1
SCHEMBL11300682 0.75 NR4A1 (0.52) NR4A1NR4A2NR4A3CDC25BMMP3
SCHEMBL30863852 0.75 NR4A1 (0.69) NR4A1NR4A2NR4A3CDC25BMMP3
SCHEMBL1600502 0.75 NR4A1 (0.69) NR4A1NR4A2NR4A3CDC25BMMP3
Naphthoic Acid SCHEMBL29352220 0.74 NR4A1 (1.00) NR4A1NR4A2NR4A3CDC25BMMP3
Naphthoic Acid SCHEMBL30233567 0.74 NR4A1 (1.00) NR4A1NR4A2NR4A3CDC25BMMP3
Naphthoic Acid SCHEMBL17258 0.74 NR4A1 (1.00) NR4A1NR4A2NR4A3CDC25BMMP3
Naphthoic Acid SCHEMBL28110155 0.74 NR4A1 (1.00) NR4A1NR4A2NR4A3CDC25BMMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2004591-A1 CYCLOPROPANES WITH CENTRAL NERVOUS SYSTEM ACTIVITY The Research Foundation Of State University Of New York (US) 2008-12-24 EP disclosed
WO-2008127223-A1 CYCLOPROPANES WITH CENTRAL NERVOUS SYSTEM ACTIVITY THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 2008-10-23 WO disclosed