SCHEMBL5047112

SCHEMBL5047112

NC(=O)CCc1ccc(CCCc2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.62
HDAC8 Q9BY41 4/20 0.59
HDAC3 O15379 3/20 0.59
HDAC2 Q92769 3/20 0.59
HDAC6 Q9UBN7 3/20 0.59
HDAC5 Q9UQL6 3/20 0.59
FFAR1 O14842 3/20 0.59
HDAC4 P56524 2/20 0.59
HDAC7 Q8WUI4 2/20 0.59
HDAC10 Q969S8 2/20 0.59
HDAC11 Q96DB2 2/20 0.59
HDAC9 Q9UKV0 2/20 0.59
MAPK1 P28482 1/20 0.59
ADRA1A P35348 1/20 0.59
SLC6A3 Q01959 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
PRMT1 Q99873 1/20 0.58
KEAP1 Q14145 1/20 0.57
HTR2A P28223 1/20 0.55
MAPT P10636 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5020712 0.92 FFAR1 (0.69) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL2593 0.92 KEAP1 (0.67) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL5020709 0.90 HDAC1 (0.67) HDAC1HDAC8HDAC3HDAC2HDAC6
Hydrazine SCHEMBL28262207 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6
Hydrochloric Acid SCHEMBL3308277 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6
Fluoride SCHEMBL27900680 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6
Ammonia Solution, Strong SCHEMBL10416110 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6
Hydrochloric Acid SCHEMBL6952080 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL7859 0.90 HDAC1 (0.72) HDAC1HDAC8HDAC3HDAC2HDAC6
Bicarbonate SCHEMBL28311766 0.90 KEAP1 (0.64) HDAC1HDAC8HDAC3HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43343-E1 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-05-01 US disclosed
EP-1233958-B1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC (CA) 2011-06-29 EP disclosed