SCHEMBL5048028

SCHEMBL5048028

O=C(O)N1CCN(C(c2ccccc2)c2ccccc2)C(CO)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
CACNA2D1 P54289 3/20 0.43
CACNA1B Q00975 3/20 0.43
CACNB1 Q02641 3/20 0.43
CACNA1H O95180 1/20 0.43
CACNA1C Q13936 1/20 0.43
KMT2A Q03164 3/20 0.43
NPC1 O15118 1/20 0.43
MAOB P27338 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
HTT P42858 1/20 0.41
USP2 O75604 1/20 0.41
MAPK1 P28482 1/20 0.41
MEN1 O00255 1/20 0.40
SLC6A9 P48067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4277413 0.83 NPC1 (0.45) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL3494682 0.83 KMT2A (0.39) CACNA2D1CACNB1KMT2AMEN1
SCHEMBL8240277 0.82 ALDH1A1 (0.41) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL4279035 0.82 GPR119 (0.44) ALDH1A1KMT2ANPC1KDM4EMAPT
SCHEMBL4283097 0.82 GRM7 (0.44) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL13701595 0.81 KMT2A (0.41) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL4275669 0.81 NPC1 (0.40) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL911824 0.80 ALDH1A1 (0.45) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1H
SCHEMBL27402706 0.80 SMN1; SMN2 (0.47) ALDH1A1KMT2AKDM4EMAPTHPGD
SCHEMBL27407208 0.80 SMN1; SMN2 (0.47) ALDH1A1KMT2AKDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976841-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2008-10-08 EP disclosed
WO-2007071035-A1 HETEROCYCLIC AMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2007-06-28 WO disclosed