SCHEMBL5049531

SCHEMBL5049531

COc1cc2nccc(Oc3ccc(NC(=O)N4CCN(c5ccccc5)C4=O)cn3)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 1.00
KDR P35968 2/20 0.64
IGF1R P08069 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5049511 0.90 MET (1.00) METKDR
SCHEMBL5094665 0.86 MET (1.00) METKDR
SCHEMBL5050781 0.84 MET (1.00) METKDRIGF1R
SCHEMBL14289201 0.83 MET (1.00) METKDR
SCHEMBL5107654 0.81 MET (1.00) METKDR
SCHEMBL5049584 0.81 MET (1.00) METKDR
SCHEMBL5056188 0.80 MET (1.00) METKDR
SCHEMBL5050783 0.80 MET (1.00) METKDR
SCHEMBL1893668 0.80 PDGFRA (0.77) METKDRIGF1R
SCHEMBL5054203 0.79 MET (1.00) METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035209-A2 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY METHYLGENE INC. (CA) 2008-03-27 WO disclosed
US-20080004273-A1 Inhibitors of protein tyrosine kinase activity METHYLGENE, INC. (CA) 2008-01-03 US disclosed
US-20080004273-A1 Inhibitors of protein tyrosine kinase activity METHYLGENE, INC. (CA) 2008-01-03 US disclosed
US-20080004273-A1 Inhibitors of protein tyrosine kinase activity METHYLGENE, INC. (CA) 2008-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004273-A1 Inhibitors of protein tyrosine kinase activity HGF, ERBB2, MET MET 3/4885KDR 11/4885IGF1R 74/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.