SCHEMBL5053765

SCHEMBL5053765

COCc1nccc2c1[nH]c1ccccc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.58
TDO2 P48775 4/20 0.58
MEN1 O00255 3/20 0.58
MAPT P10636 3/20 0.58
KMT2A Q03164 3/20 0.58
MAOA P21397 2/20 0.58
MAPK1 P28482 2/20 0.58
NPSR1 Q6W5P4 2/20 0.58
ALDH1A1 P00352 2/20 0.58
GABRP O00591 1/20 0.58
GABRD O14764 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
GABRA1 P14867 1/20 0.58
HPGD P15428 1/20 0.58
TSHR P16473 1/20 0.58
GABRB1 P18505 1/20 0.58
GABRG2 P18507 1/20 0.58
NFKB1 P19838 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1060136 0.83 TDO2 (0.63) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL11490695 0.83 KDM4E (0.71) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL28505445 0.80 DYRK1A (0.78) KDM4EMAOAALDH1A1CYP1A2CYP3A4
SCHEMBL2721049 0.80 KDM4E (0.68) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL10642447 0.79 KDM4E (0.58) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL27917573 0.77 KDM4E (0.59) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL5785176 0.77 KDM4E (0.68) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL27905044 0.77 KDM4E (0.75) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL23319492 0.76 TDO2 (0.63) KDM4ETDO2MEN1MAPTKMT2A
SCHEMBL30518089 0.76 TDO2 (0.63) KDM4ETDO2MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008132454-A1 CARBOLINES AND THEIR USE AS IMAGING AGENTS GE HEALTHCARE LIMITED (GB) 2008-11-06 WO disclosed