SCHEMBL5055185

SCHEMBL5055185

Nc1ncc(-c2ccc3c(c2)CCCN3)c(N)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.49
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
ALOX15 P16050 1/20 0.37
CASP1 P29466 1/20 0.37
HTT P42858 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
WEE1 P30291 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29114864 0.81 DHFR (0.51) DHFRADORA2AADORA1
SCHEMBL4462841 0.80 DHFR (0.56) DHFRKDM4EMAPTALDH1A1TP53
SCHEMBL9830078 0.76 DHFR (0.51) DHFRHTT
Hydrochloric Acid SCHEMBL9830813 0.75 DHFR (0.50) DHFRHTT
Hydrochloric Acid SCHEMBL30468477 0.74 ASIC3 (0.50) DHFR
SCHEMBL6555239 0.73 DHFR (0.51) DHFR
SCHEMBL30329901 0.70 DYRK1A (0.57) DHFRKDM4EMAPT
SCHEMBL8525161 0.70 MAPT (0.65) CA12CA1CA2CA9KDM4E
SCHEMBL20658532 0.70 ADORA2A (0.50) CA12CA1CA2CA9KDM4E
SCHEMBL4533554 0.70 CDK2 (0.52) KDM4EMAPTALDH1A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008079907-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY RIGEL PHARMACEUTICALS, INC. (US) 2008-07-03 WO claimed