SCHEMBL5067536

SCHEMBL5067536

O=S(=O)(Oc1cc2c(cc1CBr)CCCC2)C(F)(F)F.c1ccc(P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.33
DRD3 P35462 7/20 0.33
DRD4 P21917 5/20 0.33
DRD1 P21728 3/20 0.33
DRD5 P21918 3/20 0.33
HTR1D P28221 2/20 0.33
BRD1 O95696 1/20 0.31
BRPF1 P55201 1/20 0.31
SLC2A1 P11166 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HTR5A P47898 1/20 0.30
STS P08842 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1506497 0.89 SLC2A1 (0.36) DRD2DRD3DRD4DRD1DRD5
SCHEMBL1506583 0.76 SLC2A1 (0.39) DRD2DRD3DRD4DRD1DRD5
SCHEMBL8206659 0.73 NOTUM (0.40) KDM4EALDH1A1
SCHEMBL7107742 0.69 DRD2 (0.36) DRD2DRD3DRD4DRD1DRD5
SCHEMBL7711897 0.69 HTT (0.38) KDM4EALDH1A1
SCHEMBL12533716 0.69 STS (0.36) DRD2DRD3DRD4DRD1DRD5
SCHEMBL1506403 0.66 STS (0.34) DRD2DRD3DRD4DRD1DRD5
SCHEMBL5026108 0.66 STS (0.64) DRD2DRD3HTR1DSTSALDH1A1
SCHEMBL21468494 0.66 PTPN1 (0.40) KDM4ESTSALDH1A1
SCHEMBL10157971 0.66 DRD2 (0.34) DRD2DRD3DRD4DRD1DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1971595-A2 CETP INHIBITORS Merck & Co., Inc. (US) 2008-09-24 EP disclosed
WO-2007081569-A2 CETP INHIBITORS MERCK & CO., INC. (US) 2007-07-19 WO disclosed