SCHEMBL5067804

SCHEMBL5067804

C[C@@]1(C(=O)O)CN(C(=O)OC(I)c2ccccc2)CC1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.37
CYP2D6 P10635 5/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 2/20 0.34
OPRK1 P41145 1/20 0.34
GRIN2B Q13224 1/20 0.33
DPP4 P27487 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
ABHD6 Q9BV23 1/20 0.32
MGLL Q99685 1/20 0.32
CYP1A2 P05177 1/20 0.32
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3978561 0.84 RORC (0.38) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3975405 0.77 GRIN2B (0.44) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3976891 0.76 RORC (0.50) RORCCYP2D6CYP2C9CYP2C19GRIN2B
SCHEMBL3975897 0.73 GRIN2B (0.43) RORCCYP2D6CYP3A4GRIN2BCYP1A2
SCHEMBL4188990 0.72 CYP2D6 (0.44) CYP2D6CYP3A4OPRK1
SCHEMBL3977469 0.71 RORC (0.36) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3983521 0.71 RORC (0.36) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3976532 0.71 ALDH1A1 (0.38) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3979106 0.71 RORC (0.36) RORCCYP2D6CYP3A4CYP2C9CYP2C19
SCHEMBL3976644 0.70 ALDH1A1 (0.36) RORCCYP2D6CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1882689-A1 TRI- OR TETRA-SUBSTITUTED-3-AMINOPYRROLIDINE DERIVATIVES Daiichi Sankyo Company, Limited (JP) 2008-01-30 EP disclosed