SCHEMBL5068474

SCHEMBL5068474

C=CC(=O)OCc1ccc(CC)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.49
TSHR P16473 6/20 0.44
HPGD P15428 1/20 0.44
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
HCAR2 Q8TDS4 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 6/20 0.42
NAAA Q02083 1/20 0.42
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 2/20 0.39
HIF1A Q16665 2/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2556244 0.90 HCAR2 (0.50) THRBTSHRHPGDHCAR2MEN1
SCHEMBL12149338 0.88 THRB (0.40) THRBTSHRHPGDRXRARXRB
SCHEMBL13783953 0.86 THRB (0.68) THRBTSHRHPGDHCAR2MEN1
SCHEMBL149067 0.85 MMP2 (0.45) THRBHCAR2ALDH1A1NAAAMAPT
SCHEMBL9419668 0.85 TSHR (0.47) THRBTSHRHPGDHCAR2MEN1
SCHEMBL17791314 0.85 THRB (0.51) THRBTSHRHCAR2MEN1KMT2A
SCHEMBL16125662 0.85 HCAR2 (0.46) THRBTSHRHPGDHCAR2MEN1
SCHEMBL12367978 0.85 HCAR2 (0.46) THRBTSHRHPGDHCAR2MEN1
SCHEMBL12268165 0.85 HCAR2 (0.46) THRBTSHRHPGDHCAR2MEN1
SCHEMBL4578050 0.85 MEN1 (0.55) THRBTSHRHCAR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4479101-B1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUE COHESIVES (FR) 2026-03-04 EP claimed
US-20250170299-A1 SURGICAL ADHESIVES COHESIVES (FR) 2025-05-29 US claimed
US-20250152772-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUES COHESIVES (FR) 2025-05-15 US claimed
US-12239759-B2 Surgical adhesives COHESIVES (FR) 2025-03-04 US claimed
EP-4479101-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUE Cohesives (FR) 2024-12-25 EP claimed
WO-2023156749-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUE COHESIVES (FR) 2023-08-24 WO claimed
US-20220143264-A1 SURGICAL ADHESIVES COHESIVES (FR) 2022-05-12 US claimed
US-11207443-B2 Surgical adhesives COHESIVES (FR) 2021-12-28 US claimed
US-20180280564-A1 SURGICAL ADHESIVES COHESIVES (FR) 2018-10-04 US claimed
EP-1015505-B1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE INC (US) 2005-03-09 EP claimed
EP-0783710-B1 POLYESTER RESIN-BASED HIGH INDEX OPHTHALMIC LENSES HAVING IMPROVED OPTICAL UNIFORMITY AND/OR TINTABILITY SIGNET ARMORLITE INC (US) 2002-05-29 EP claimed
US-6099123-A A CROSSLINKABLE CASTING POLYMERIC MATERIAL CONSISTS OF AN UNSATURATED POLYESTER, A CROSSLINKING AGENT AND A PHOTOINITIATORS SIGNET ARMORLITE, INC. (US) 2000-08-08 US claimed
EP-1015505-A1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE, INC. (US) 2000-07-05 EP claimed
US-5886764-A UNSATURATED POLYESTER RESIN, AN ADDITIVE SELECTED FROM THE GROUP CONSISTING OF ABOUT 1% TO ABOUT 20% BY WEIGHT OF AN ALLYLIC ESTER MONOMER, ABOUT 1% TO ABOUT 20% BY WEIGHT OF AN ACRYLATE, AND MIXTURES THEREOF, AND AN EXOTHERM DEPRESSANT SIGNET ARMORLITE, INC. (US) 1999-03-23 US claimed
WO-1999011682-A1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE, INC. (US) 1999-03-11 WO claimed
US-5852112-A Polyester resin-based high index ophthalmic lenses having improved optical unformity and/or tintability SIGNET ARMORLITE, INC. (US) 1998-12-22 US claimed
US-5694195-A Polyester resin-based high index ophthalmic lenses having improved optical uniformity and/or tintability SIGNET ARMORLITE, INC. (US) 1997-12-02 US claimed
EP-0783710-A1 POLYESTER RESIN-BASED HIGH INDEX OPHTHALMIC LENSES HAVING IMPROVED OPTICAL UNIFORMITY AND/OR TINTABILITY SIGNET ARMORLITE, INC. (US) 1997-07-16 EP claimed
WO-1996010760-A1 POLYESTER RESIN-BASED HIGH INDEX OPHTHALMIC LENSES HAVING IMPROVED OPTICAL UNIFORMITY AND/OR TINTABILITY SIGNET ARMORLITE, INC. (US) 1996-04-11 WO claimed
US-20250170299-A1 SURGICAL ADHESIVES COHESIVES (FR) 2025-05-29 US disclosed
US-20250152772-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUES COHESIVES (FR) 2025-05-15 US disclosed
US-12239759-B2 Surgical adhesives COHESIVES (FR) 2025-03-04 US disclosed
EP-4479101-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUE Cohesives (FR) 2024-12-25 EP disclosed
WO-2023156749-A1 PHOTOPOLYMERISABLE COMPOSITION FOR ADHESIVE FOR BIOLOGICAL TISSUE COHESIVES (FR) 2023-08-24 WO disclosed
US-20220143264-A1 SURGICAL ADHESIVES COHESIVES (FR) 2022-05-12 US disclosed
EP-3297692-B1 SURGICAL ADHESIVES COHESIVES (FR) 2022-01-05 EP disclosed
US-11207443-B2 Surgical adhesives COHESIVES (FR) 2021-12-28 US disclosed
CN-107771086-B Surgical adhesive 寇希西弗斯公司 2021-11-05 CN disclosed
WO-2020059668-A1 PIGMENT-CONTAINING RESIN COMPOSITION 花王株式会社 2020-03-26 WO disclosed
US-20180280564-A1 SURGICAL ADHESIVES COHESIVES (FR) 2018-10-04 US disclosed
US-9599760-B2 Composition for optical film, and films and display device SAMSUNG ELECTRONICS CO., LTD. (KR) 2017-03-21 US disclosed
US-9441065-B2 Curable composition for imprints, cured product and method for manufacturing a cured product FUJIFILM CORPORATION (JP) 2016-09-13 US disclosed
US-9441065-B2 Curable composition for imprints, cured product and method for manufacturing a cured product FUJIFILM CORPORATION (JP) 2016-09-13 US disclosed
US-8999221-B2 Curable composition for imprints, patterning method and pattern FUJIFILM CORPORATION (JP) 2015-04-07 US disclosed
US-8999221-B2 Curable composition for imprints, patterning method and pattern FUJIFILM CORPORATION (JP) 2015-04-07 US disclosed
US-8883065-B2 Curable composition for imprints, patterning method and pattern FUJIFILM CORPORATION (JP) 2014-11-11 US disclosed
US-8883065-B2 Curable composition for imprints, patterning method and pattern FUJIFILM CORPORATION (JP) 2014-11-11 US disclosed
US-20140121292-A1 CURABLE COMPOSITION FOR IMPRINTS, PATTERNING METHOD AND PATTERN FUJIFILM CORPORATION (JP) 2014-05-01 US disclosed
US-20140121292-A1 CURABLE COMPOSITION FOR IMPRINTS, PATTERNING METHOD AND PATTERN FUJIFILM CORPORATION (JP) 2014-05-01 US disclosed
US-20110236595-A1 CURABLE COMPOSITION FOR IMPRINTS, PATTERNING METHOD AND PATTERN FUJIFILM CORPORATION (JP) 2011-09-29 US disclosed
US-20110236595-A1 CURABLE COMPOSITION FOR IMPRINTS, PATTERNING METHOD AND PATTERN FUJIFILM CORPORATION (JP) 2011-09-29 US disclosed
EP-1549483-B1 METHODS FOR PREPARING COMPOSITE PHOTOCHROMIC OPHTHALMIC LENSES AND A PHOTOCHROMIC LENS & xA; SIGNET ARMORLITE INC (US) 2008-04-16 EP disclosed
US-7273911-B2 Self-adhesive addition-crosslinking silicone compositions WACKER CHEMIE AG (DE) 2007-09-25 US disclosed
US-7119159-B2 Self-adhesive addition-crosslinking silicon compositions WACKER-CHEMIE GMBH (DE) 2006-10-10 US disclosed
EP-1015505-B1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE INC (US) 2005-03-09 EP disclosed
US-6863848-B2 Methods for preparing composite photochromic ophthalmic lenses SIGNET ARMORLITE, INC. (US) 2005-03-08 US disclosed
US-20050042462-A1 Self-adhesive addition-crosslinking silicone compositions WACKER-CHEMIE GMBH (DE) 2005-02-24 US disclosed
US-6790533-B2 BLEND OF POLYSILOXANE AND FILLER WACKER-CHEMIE GMBH (DE) 2004-09-14 US disclosed
US-20040041287-A1 Methods for preparing composite photochromic ophthalmic lenses SIGNET ARMORLITE, INC. 2004-03-04 US disclosed
US-20030236380-A1 Self-adhesive addition-crosslinking silicon compositions WACKER-CHEMIE GMBH (DE) 2003-12-25 US disclosed
US-20020187358-A1 Self-adhesive thermally crosslinkable 1-component silicone compositions WACKER-CHEMIE GMBH (DE) 2002-12-12 US disclosed
EP-0783710-B1 POLYESTER RESIN-BASED HIGH INDEX OPHTHALMIC LENSES HAVING IMPROVED OPTICAL UNIFORMITY AND/OR TINTABILITY SIGNET ARMORLITE INC (US) 2002-05-29 EP disclosed
US-6099123-A A CROSSLINKABLE CASTING POLYMERIC MATERIAL CONSISTS OF AN UNSATURATED POLYESTER, A CROSSLINKING AGENT AND A PHOTOINITIATORS SIGNET ARMORLITE, INC. (US) 2000-08-08 US disclosed
EP-1015505-A1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE, INC. (US) 2000-07-05 EP disclosed
US-5886764-A UNSATURATED POLYESTER RESIN, AN ADDITIVE SELECTED FROM THE GROUP CONSISTING OF ABOUT 1% TO ABOUT 20% BY WEIGHT OF AN ALLYLIC ESTER MONOMER, ABOUT 1% TO ABOUT 20% BY WEIGHT OF AN ACRYLATE, AND MIXTURES THEREOF, AND AN EXOTHERM DEPRESSANT SIGNET ARMORLITE, INC. (US) 1999-03-23 US disclosed
WO-1999011682-A1 PRODUCTION OF PHOTOPOLYMERIZED POLYESTER HIGH INDEX OPHTHALMIC LENSES SIGNET ARMORLITE, INC. (US) 1999-03-11 WO disclosed
US-5852112-A Polyester resin-based high index ophthalmic lenses having improved optical unformity and/or tintability SIGNET ARMORLITE, INC. (US) 1998-12-22 US disclosed
US-5694195-A Polyester resin-based high index ophthalmic lenses having improved optical uniformity and/or tintability SIGNET ARMORLITE, INC. (US) 1997-12-02 US disclosed
US-5694195-A Polyester resin-based high index ophthalmic lenses having improved optical uniformity and/or tintability SIGNET ARMORLITE, INC. (US) 1997-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110236595-A1 CURABLE COMPOSITION FOR IMPRINTS, PATTERNING METHOD AND PATTERN DNMT3L, DNMT3A, DNMT1 THRB 3880/4885TSHR 4211/4885HPGD 4554/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.